@article{UBHD-69232236, author={Chen, Xin and Chen, Xinyang and Steimbach, Raphael R. and Wu, Tong and Li, Hongmei and Dan, Wenjia and Shi, Peidong and Cao, Chenyu and Li, Ding and Miller, Aubry K. and Qiu, Zhixia and Gao, Jinming and Zhu, Yong}, title={Novel 2, 5-diketopiperazine derivatives as potent selective histone deacetylase 6 inhibitors}, subtitle={rational design, synthesis and antiproliferative activity}, year={2020}, pages={1-13}, language={eng}, issn={1768-3254}, volume={187}, number={Artikel-ID 111950}, note={Gesehen am 10.07.2024}, journal={European journal of medicinal chemistry}, doi={10.1016/j.ejmech.2019.111950}, } @article{UBHD-68648949, author={Herbst-Gervasoni, Corey J. and Steimbach, Raphael R. and Morgen, Michael and Miller, Aubry K. and Christianson, David W.}, title={Structural basis for the selective inhibition of HDAC10, the cytosolic polyamine deacetylase}, year={2020}, pages={2154-2163}, language={eng}, issn={1554-8937}, volume={15}, number={8}, note={Gesehen am 15.10.2020}, journal={ACS chemical biology}, doi={10.1021/acschembio.0c00362}, } @article{UBHD-69081323, author={Herp, Daniel and Ridinger, Johannes and Robaa, Dina and Shinsky, Stephen A. and Schmidtkunz, Karin and Yesiloglu, Talha Z. and Bayer, Theresa Yasmin Charlotte and Steimbach, Raphael R. and Herbst-Gervasoni, Corey J. and Merz, Annika and Romier, Christophe and Sehr, Peter and Gunkel, Nikolas and Miller, Aubry K. and Christianson, David W. and Oehme, Ina and Sippl, Wolfgang and Jung, Manfred}, title={First fluorescent acetylspermidine deacetylation assay for HDAC10 identifies selective inhibitors with cellular target engagement}, year={2022}, pages={1-28}, language={eng}, issn={1439-7633}, volume={23}, note={Published online: 24 May 2022}, journal={ChemBioChem}, doi={10.1002/cbic.202200180}, } @article{UBHD-69232142, author={Lechner, Severin and Malgapo, Martin Ian P. and Gr{\"a}tz, Christian and Steimbach, Raphael R. and Baron, Agnes and R{\"u}ther, Patrick and Nadal, Simon and Stumpf, Carmen and Loos, Christina and Ku, Xin and Prokofeva, Polina and Lautenbacher, Ludwig and Heimburg, Tino and W{\"u}rf, Vivian and Meng, Chen and Wilhelm, Mathias and Sippl, Wolfgang and Kleigrewe, Karin and Pauling, Josch K. and Kramer, Karl and Miller, Aubry K. and Pfaffl, Michael W. and Linder, Maurine E. and K{\"u}ster, Bernhard and Médard, Guillaume}, title={Author correction: Target deconvolution of HDAC pharmacopoeia reveals MBLAC2 as common off-target}, year={2022}, pages={1}, language={eng}, issn={1552-4469}, volume={18}, number={Artikel-ID 913}, journal={Nature chemical biology}, doi={10.1038/s41589-022-01112-5}, } @article{UBHD-69135636, author={Lechner, Severin and Steimbach, Raphael R. and Wang, Longlong and Deline, Marshall L. and Chang, Yun-Chien and Fromme, Tobias and Klingenspor, Martin and Matthias, Patrick and Miller, Aubry K. and Médard, Guillaume and Kuster, Bernhard}, title={Chemoproteomic target deconvolution reveals Histone Deacetylases as targets of (R)-lipoic acid}, year={2023}, pages={1-10}, language={eng}, issn={2041-1723}, volume={14}, number={Artikel-ID 3548}, note={Gesehen am 31.10.2023}, journal={Nature Communications}, doi={10.1038/s41467-023-39151-8}, } @article{UBHD-69081322, author={Lechner, Severin and Malgapo, Martin Ian P. and Gr{\"a}tz, Christian and Steimbach, Raphael R. and Baron, Agnes and R{\"u}ther, Patrick and Nadal, Simon and Stumpf, Carmen and Loos, Christina and Ku, Xin and Prokofeva, Polina and Lautenbacher, Ludwig and Heimburg, Tino and W{\"u}rf, Vivian and Meng, Chen and Wilhelm, Mathias and Sippl, Wolfgang and Kleigrewe, Karin and Pauling, Josch K. and Kramer, Karl and Miller, Aubry K. and Pfaffl, Michael W. and Linder, Maurine E. and Kuster, Bernhard and Médard, Guillaume}, title={Target deconvolution of HDAC pharmacopoeia reveals MBLAC2 as common off-target}, year={2022}, pages={812-820}, language={eng}, issn={1552-4469}, volume={18}, journal={Nature chemical biology}, doi={10.1038/s41589-022-01015-5}, } @article{UBHD-69287942, author={Liang, Ting and Liu, Shiru and Dang, Baiyun and Luan, Xiaofa and Guo, Yifan and Steimbach, Raphael R. and Hu, Jiadong and Lu, Long and Yue, Peiyu and Wang, Ruotian and Zheng, Meng and Gao, Jinming and Yin, Xia and Chen, Xin}, title={Multimechanism biological profiling of tetrahydro-β-carboline analogues as selective HDAC6 inhibitors for the treatment of Alzheimer's disease}, year={2024}, pages={1-18}, language={eng}, issn={1768-3254}, volume={275(2024) vom: Sept.}, number={Artikel-ID 116624}, note={Online verf{\"u}gbar 24 June 2024, Version des Artikel 25 June 2024 ; Gesehen am 08.01.2025}, journal={European journal of medicinal chemistry}, doi={10.1016/j.ejmech.2024.116624}, } @article{UBHD-68881016, author={Steimbach, Raphael R. and Tihanyi, Gergely and Géraldy, Magalie N. E. and Wzorek, Alicja and Miller, Aubry K. and Klika, Karel D.}, title={Can an intermediate rate of nitrogen inversion affect drug efficacy?}, year={2021}, pages={1-14}, language={eng}, issn={2073-8994}, volume={13}, note={Gesehen am 21.02.2022}, journal={Symmetry}, doi={10.3390/sym13091753}, } @book{UBHD-69081046, author={Steimbach, Raphael R.}, organization={Universit{\"a}t Heidelberg}, title={Selective inhibitors and targeted degraders of histone deacetylase 10}, address={Heidelberg}, year={2023}, pages={455 Seiten}, language={eng}, school={Dissertation, Ruprecht-Karls-University Heidelberg, 2023}, library={UB [Signatur: 2023 U 437]}, } @book{UBHD-69164348, author={Steimbach, Raphael R.}, title={Selective inhibitors and targeted degraders of histone deacetylase 10}, address={Heidelberg}, year={2023}, pages={1 Online-Ressource (461 Seiten)}, language={eng}, school={Dissertation, Ruprecht-Karls-University Heidelberg, 2023}, doi={10.11588/heidok.00033158}, url={https://nbn-resolving.org/urn:nbn:de:bsz:16-heidok-331582}, library={UB}, }